Nielsen TE, Schreiber SL. Towards the optimal screening collection: a synthesis strategy. Angew Chem Int Ed Engl. 2008;47(1):48-56. doi:10.1002/anie.200703073
Fitzgerald ME, Mulrooney CA, Duvall JR, et al. Build/couple/pair strategy for the synthesis of stereochemically diverse macrolactams via head-to-tail cyclization. ACS Comb Sci. 2012;14(2):89-96. doi:10.1021/co200161z
Lowe JT, Lee MD, Akella LB, et al. Synthesis and profiling of a diverse collection of azetidine-based scaffolds for the development of CNS-focused lead-like libraries. J Org Chem. 2012;77(17):7187-211. doi:10.1021/jo300974j
Gerard B, O’Shea MW, Donckele E, et al. Application of a catalytic asymmetric Povarov reaction using chiral ureas to the synthesis of a tetrahydroquinoline library. ACS Comb Sci. 2012;14(11):621-30. doi:10.1021/co300098v
Wang Y, Jimenez M, Sheehan P, et al. Selective access to trisubstituted macrocyclic E- and Z-alkenes from the ring-closing metathesis of vinylsiloxanes. Org Lett. 2013;15(6):1218-21. doi:10.1021/ol400134d
Gerard B, Lee MD, Dandapani S, et al. Synthesis of stereochemically and skeletally diverse fused ring systems from functionalized C-glycosides. J Org Chem. 2013;78(11):5160-71. doi:10.1021/jo4000916
Nelson SD, Wawer MJ, Schreiber SL. Divergent Synthesis and Real-Time Biological Annotation of Optically Active Tetrahydrocyclopenta[c]pyranone Derivatives. Org Lett. 2016;18(24):6280-6283. doi:10.1021/acs.orglett.6b03118